- Source: AM-2233
AM-2233 is a drug that acts as a highly potent full agonist for the cannabinoid receptors, with a Ki of 1.8 nM at CB1 and 2.2 nM at CB2 as the active (R) enantiomer. It was developed as a selective radioligand for the cannabinoid receptors and has been used as its 131I derivative for mapping the distribution of the CB1 receptor in the brain. AM-2233 was found to fully substitute for THC in rats, with a potency lower than that of JWH-018 but higher than WIN 55,212-2.
It is notable for inducing tinnitus, though the reasons for this are unclear and may provide valuable insight into tinnitus research.
Legal Status
As of October 2015 AM-2233 is a controlled substance in China.
See also
AM-679
AM-694
AM-1220
AM-1221
AM-1235
AM-1241
AM-2232
Cannabipiperidiethanone
FUBIMINA
JWH-018
List of AM cannabinoids
List of JWH cannabinoids
List of HU cannabinoids
List of designer drugs
References
Kata Kunci Pencarian:
- Pembagian administratif Timor Leste
- Unsur golongan 4
- Nikotinamida adenina dinukleotida
- Daftar bintang di rasi bintang Vela
- Daftar planet minor: 52001–53000
- Daftar planet minor: 65001–66000
- Daftar bintang di rasi bintang Sagittarius
- Hafnium
- Daftar Minuscule Perjanjian Baru (2001–)
- AM-2233
- AM-2201
- Psilocybe cubensis
- Ayahuasca
- Synthetic cannabinoids
- 1S-LSD
- Tetrahydrocannabiphorol
- Morning glory
- Dimethylheptylpyran
- Tetrahydrocannabinolic acid
