- Source: List of adrenergic drugs
This is a list of adrenergic drugs. These are pharmaceutical drugs, naturally occurring compounds and other chemicals that influence the function of the neurotransmitter epinephrine (adrenaline).
Receptor ligands
= α1-adrenergic receptor ligands
=Agonists
Antagonists
Many tricyclic antidepressants, tetracyclic antidepressants, antipsychotics, ergolines, and some piperazines like buspirone, trazodone, nefazodone, etoperidone, and mepiprazole antagonize α1-adrenergic receptors as well, which contributes to their side effects such as orthostatic hypotension.
= α2-adrenergic receptor ligands
=Agonists
Antagonists
Many atypical antipsychotics and azapirones like buspirone and gepirone (via metabolite pyrimidinylpiperazine) antagonize α2-adrenergic receptors as well.
= β-adrenergic receptor ligands
=Agonists
Antagonists
Reuptake inhibitors
= Norepinephrine transporter (NET) inhibitors
== Vesicular monoamine transporter (VMAT) inhibitors
=Releasing agents
Enzyme inhibitors
= Anabolism
=Phenylalanine hydroxylase (PAH) inhibitors
Tyrosine hydroxylase inhibitors
Aromatic L-amino acid decarboxylase (AAAD) inhibitors
Dopamine-beta-hydroxylase (DBH) inhibitors
Phenylethanolamine N-methyltransferase (PNMT) inhibitors
= Catabolism
=Monoamine oxidase (MAO) inhibitors
MAO-B inhibitors also influence norepinephrine/epinephrine levels since they inhibit the breakdown of their precursor dopamine.
Catechol-O-methyl transferase (COMT) inhibitors
Others
= Precursors
== Cofactors
== Activity enhancers
== Release blockers
== Toxins
=References
Kata Kunci Pencarian:
- Antipiretik
- Efedrin
- Metoprolol
- Reseptor terhubung protein G
- Metilfenidat
- Diabetes melitus
- Teofilin/efedrin
- Antihipertensi
- List of adrenergic drugs
- Adrenergic agonist
- Adrenergic
- Adrenergic antagonist
- Norepinephrine reuptake inhibitor
- List of veterinary drugs
- Alpha-2 adrenergic receptor
- Adrenergic blocking agent
- Beta-2 adrenergic receptor
- Beta-adrenergic agonist
